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CCOC(=O)N1CCC(C(=O)Nc2ccc(NC(=O)N3CCC(C(=O)OCC(F)(F)F)CC3)cc2)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000453 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A017742 | PGDB_C019884 | PGDB_AS002246 | View | |
| Dmax | - | = | 2.82 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A024085 | PGDB_C019884 | PGDB_AS000856 | View | |
| Dmax | - | = | 15.52 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A027215 | PGDB_C019884 | PGDB_AS001280 | View | |
| EC50 | - | = | 0.0000000074 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A037118 | PGDB_C019884 | PGDB_AS002126 | View | |
| Dmax | - | = | 1.76 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A045955 | PGDB_C019884 | PGDB_AS000546 | View | |
| EC50 | - | = | 0.000000000298 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A046502 | PGDB_C019884 | PGDB_AS001078 | View | |
| EC50 | - | = | 0.0000453 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A063819 | PGDB_C019884 | PGDB_AS001009 | View | |
| EC50 | - | = | 0.0000096 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A063830 | PGDB_C019884 | PGDB_AS000046 | View | |
| EC50 | - | = | 0.0000453 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A073951 | PGDB_C019884 | PGDB_AS001381 | View |