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Compound
PGDB_C019885
9 activity records1 related patents
2D structure
CC(=O)Nc1ccc(NC(=O)Cn2cnc3c(cnn3C(C)(C)C)c2=O)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000134 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A009964 | PGDB_C019885 | PGDB_AS000046 | View |
| Dmax | - | = | 0.27 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A015801 | PGDB_C019885 | PGDB_AS000856 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A033733 | PGDB_C019885 | PGDB_AS001381 | View |
| Dmax | - | = | 0.23 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A042494 | PGDB_C019885 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000000182 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A048490 | PGDB_C019885 | PGDB_AS002126 | View |
| Dmax | - | = | 15.16 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A055738 | PGDB_C019885 | PGDB_AS001280 | View |
| EC50 | - | = | 0.0000305 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A056583 | PGDB_C019885 | PGDB_AS001078 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A069174 | PGDB_C019885 | PGDB_AS001009 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A070420 | PGDB_C019885 | PGDB_AS002246 | View |