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Compound
PGDB_C019887
9 activity records1 related patents
2D structure
O=C(c1ccco1)N1CCN(c2ncc(-c3cccc(NC(=O)C(F)(F)F)c3)n3ccnc23)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000000203 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A008602 | PGDB_C019887 | PGDB_AS002126 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A014448 | PGDB_C019887 | PGDB_AS001381 | View |
| Dmax | - | = | 1.97 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A017928 | PGDB_C019887 | PGDB_AS000856 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A021925 | PGDB_C019887 | PGDB_AS002246 | View |
| Dmax | - | = | 14.24 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A030042 | PGDB_C019887 | PGDB_AS001280 | View |
| EC50 | - | = | 0.0000215 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A032146 | PGDB_C019887 | PGDB_AS001078 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A037050 | PGDB_C019887 | PGDB_AS001009 | View |
| Dmax | - | = | 1.06 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A063141 | PGDB_C019887 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000165 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A076788 | PGDB_C019887 | PGDB_AS000046 | View |