Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C019888
9 activity records1 related patents
2D structure
CCN(CC)c1ccc2cc(-c3nc(C)cs3)c(=O)oc2c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A010673 | PGDB_C019888 | PGDB_AS002246 | View |
| EC50 | - | = | 0.0000116 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A014099 | PGDB_C019888 | PGDB_AS002126 | View |
| Dmax | - | = | 13.93 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A015448 | PGDB_C019888 | PGDB_AS001280 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A015612 | PGDB_C019888 | PGDB_AS001009 | View |
| EC50 | - | = | 0.0000082 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A049029 | PGDB_C019888 | PGDB_AS000046 | View |
| Dmax | - | = | 6.67 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A049719 | PGDB_C019888 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000168 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A052982 | PGDB_C019888 | PGDB_AS001078 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A060422 | PGDB_C019888 | PGDB_AS001381 | View |
| Dmax | - | = | 0.77 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A067740 | PGDB_C019888 | PGDB_AS000856 | View |