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Compound
PGDB_C019889
9 activity records1 related patents
2D structure
CCN(CC)c1ccc2c(c1)OC(N)=C(C#N)C2c1ccccc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A008738 | PGDB_C019889 | PGDB_AS001009 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A032529 | PGDB_C019889 | PGDB_AS002246 | View |
| EC50 | - | = | 0.0000314 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A039058 | PGDB_C019889 | PGDB_AS000046 | View |
| Dmax | - | = | 0.22 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A046487 | PGDB_C019889 | PGDB_AS000856 | View |
| EC50 | - | = | 0.0000125 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A047737 | PGDB_C019889 | PGDB_AS001078 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A049868 | PGDB_C019889 | PGDB_AS001381 | View |
| EC50 | - | = | 0.0000754 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A057965 | PGDB_C019889 | PGDB_AS002126 | View |
| Dmax | - | = | 6.24 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A069673 | PGDB_C019889 | PGDB_AS000546 | View |
| Dmax | - | = | 13.74 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A069938 | PGDB_C019889 | PGDB_AS001280 | View |