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CCOC(=O)C1=CN(Cc2ccc(OC)cc2)C=C(C(=O)OCC)C1c1ccccc1OCc1ccccc1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000442 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A013409 | PGDB_C019891 | PGDB_AS001009 | View | |
| Dmax | - | = | 3.64 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A021801 | PGDB_C019891 | PGDB_AS000546 | View | |
| Dmax | - | = | 2.45 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A022143 | PGDB_C019891 | PGDB_AS000856 | View | |
| EC50 | - | = | 0.0000157 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A034072 | PGDB_C019891 | PGDB_AS002126 | View | |
| EC50 | - | = | 0.0000000062 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A035906 | PGDB_C019891 | PGDB_AS001078 | View | |
| EC50 | - | = | 0.0000442 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A046742 | PGDB_C019891 | PGDB_AS001381 | View | |
| EC50 | - | = | 0.0000161 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A050778 | PGDB_C019891 | PGDB_AS000046 | View | |
| EC50 | - | = | 0.0000442 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A054041 | PGDB_C019891 | PGDB_AS002246 | View | |
| Dmax | - | = | 11.97 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A073130 | PGDB_C019891 | PGDB_AS001280 | View |