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Compound
PGDB_C019892
9 activity records1 related patents
2D structure
O=C(CCc1nc(-c2ccncc2)no1)N1CCN(c2cccc(C(F)(F)F)c2)C(C(F)(F)F)C1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A029807 | PGDB_C019892 | PGDB_AS001009 | View |
| EC50 | - | = | 0.0000000253 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A032584 | PGDB_C019892 | PGDB_AS001078 | View |
| EC50 | - | = | 0.0000109 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A035491 | PGDB_C019892 | PGDB_AS002126 | View |
| Dmax | - | = | -0.2133 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A048695 | PGDB_C019892 | PGDB_AS000546 | View |
| Dmax | - | = | 0.31 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A058359 | PGDB_C019892 | PGDB_AS000856 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A058989 | PGDB_C019892 | PGDB_AS001381 | View |
| Dmax | - | = | 10.2 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A063360 | PGDB_C019892 | PGDB_AS001280 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A073396 | PGDB_C019892 | PGDB_AS002246 | View |
| EC50 | - | = | 0.0000106 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A076092 | PGDB_C019892 | PGDB_AS000046 | View |