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CCOC(=O)c1sc2ncn(CC(=O)NCCC3=CCCCC3)c(=O)c2c1C| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A022126 | PGDB_C019893 | PGDB_AS001381 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A023680 | PGDB_C019893 | PGDB_AS001009 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A027291 | PGDB_C019893 | PGDB_AS002246 | View | |
| Dmax | - | = | 10.3 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A027401 | PGDB_C019893 | PGDB_AS001280 | View | |
| EC50 | - | = | 0.0000000478 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A029606 | PGDB_C019893 | PGDB_AS001078 | View | |
| Dmax | - | = | 0.7 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A037587 | PGDB_C019893 | PGDB_AS000546 | View | |
| EC50 | - | = | 0.0000001376 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A040638 | PGDB_C019893 | PGDB_AS002126 | View | |
| EC50 | - | = | 0.0000014 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A060535 | PGDB_C019893 | PGDB_AS000046 | View | |
| Dmax | - | = | 0.13 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A061621 | PGDB_C019893 | PGDB_AS000856 | View |