Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C019895
9 activity records1 related patents
2D structure
COc1cc(C)c(C)cc1N1C(=O)c2ccc(C(=O)Nc3cc([N+](=O)[O-])ccc3O)cc2C1=OCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000000089 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A007025 | PGDB_C019895 | PGDB_AS001078 | View |
| EC50 | - | = | 0.0000221 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A014471 | PGDB_C019895 | PGDB_AS000046 | View |
| EC50 | - | = | 0.0000212 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A024689 | PGDB_C019895 | PGDB_AS002126 | View |
| Dmax | - | = | 2.25 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A035723 | PGDB_C019895 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A039830 | PGDB_C019895 | PGDB_AS001009 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A044915 | PGDB_C019895 | PGDB_AS001381 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A045248 | PGDB_C019895 | PGDB_AS002246 | View |
| Dmax | - | = | 10.59 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A052786 | PGDB_C019895 | PGDB_AS001280 | View |
| Dmax | - | = | 0.49 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A075823 | PGDB_C019895 | PGDB_AS000856 | View |