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Compound
PGDB_C019896
9 activity records1 related patents
2D structure
Cc1ccc2nc(SCC(=O)Nc3ncc(C)s3)c(C#N)cc2c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A007624 | PGDB_C019896 | PGDB_AS001009 | View |
| EC50 | - | = | 0.0000000000228 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A009635 | PGDB_C019896 | PGDB_AS001078 | View |
| Dmax | - | = | 0.24 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A014199 | PGDB_C019896 | PGDB_AS000856 | View |
| Dmax | - | = | 10.71 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A020802 | PGDB_C019896 | PGDB_AS001280 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A035041 | PGDB_C019896 | PGDB_AS002246 | View |
| EC50 | - | = | 0.0000149 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A043644 | PGDB_C019896 | PGDB_AS000046 | View |
| Dmax | - | = | 35.62 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A051899 | PGDB_C019896 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000162 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A063387 | PGDB_C019896 | PGDB_AS002126 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A076787 | PGDB_C019896 | PGDB_AS001381 | View |