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Compound
PGDB_C019897
9 activity records1 related patents
2D structure
COc1ccc(NC(=O)c2cc(S(=O)(=O)N3CCN(c4ccc(C)cn4)CC3)ccc2F)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000000032 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A007727 | PGDB_C019897 | PGDB_AS000046 | View |
| EC50 | - | = | 0.0000000002416 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A026765 | PGDB_C019897 | PGDB_AS001078 | View |
| EC50 | - | = | 0.0000546 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A033194 | PGDB_C019897 | PGDB_AS001009 | View |
| EC50 | - | = | 0.0000546 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A036809 | PGDB_C019897 | PGDB_AS002246 | View |
| EC50 | - | = | 0.0000000002173 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A050289 | PGDB_C019897 | PGDB_AS002126 | View |
| Dmax | - | = | 1.99 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A060322 | PGDB_C019897 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000546 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A061874 | PGDB_C019897 | PGDB_AS001381 | View |
| Dmax | - | = | 11.58 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A063706 | PGDB_C019897 | PGDB_AS001280 | View |
| Dmax | - | = | 2.43 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A064178 | PGDB_C019897 | PGDB_AS000856 | View |