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COc1ccc(SCC(=O)NNC(=S)Nc2ccccc2)cc1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 10.12 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A012242 | PGDB_C019898 | PGDB_AS001280 | View | |
| EC50 | - | = | 0.0000000005406 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A014429 | PGDB_C019898 | PGDB_AS001078 | View | |
| Dmax | - | = | 2.8 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A018479 | PGDB_C019898 | PGDB_AS000856 | View | |
| EC50 | - | = | 0.0000566 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A018497 | PGDB_C019898 | PGDB_AS001009 | View | |
| EC50 | - | = | 0.0000000075 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A033065 | PGDB_C019898 | PGDB_AS002126 | View | |
| EC50 | - | = | 0.0000073 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A037207 | PGDB_C019898 | PGDB_AS000046 | View | |
| EC50 | - | = | 0.0000566 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A038018 | PGDB_C019898 | PGDB_AS001381 | View | |
| Dmax | - | = | 2.56 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A056194 | PGDB_C019898 | PGDB_AS000546 | View | |
| EC50 | - | = | 0.0000566 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A065179 | PGDB_C019898 | PGDB_AS002246 | View |