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CCC(C)OC(=O)C1=C(C)NC2=C(C(=O)CC(c3ccc(F)cc3)C2)C1c1cccc(Cl)c1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000241 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A009333 | PGDB_C019900 | PGDB_AS002126 | View | |
| Dmax | - | = | 0.13 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A024979 | PGDB_C019900 | PGDB_AS000856 | View | |
| EC50 | - | = | 0.0000221 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A028055 | PGDB_C019900 | PGDB_AS001078 | View | |
| Dmax | - | = | 4.29 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A039161 | PGDB_C019900 | PGDB_AS000546 | View | |
| EC50 | - | = | 0.0000458 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A041224 | PGDB_C019900 | PGDB_AS001381 | View | |
| EC50 | - | = | 0.0000458 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A048513 | PGDB_C019900 | PGDB_AS001009 | View | |
| EC50 | - | = | 0.0000458 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A050154 | PGDB_C019900 | PGDB_AS002246 | View | |
| EC50 | - | = | 0.000016 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A070234 | PGDB_C019900 | PGDB_AS000046 | View | |
| Dmax | - | = | 9.85 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A076901 | PGDB_C019900 | PGDB_AS001280 | View |