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Compound
PGDB_C019903
9 activity records1 related patents
2D structure
COc1ccc(COC(=O)C2=C(C)NC3=C(C(=O)CC(C)(C)C3)C2c2ccccc2)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000238 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A009365 | PGDB_C019903 | PGDB_AS000046 | View |
| Dmax | - | = | 1.77 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A013592 | PGDB_C019903 | PGDB_AS000856 | View |
| EC50 | - | = | 0.0000000072 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A022783 | PGDB_C019903 | PGDB_AS001078 | View |
| EC50 | - | = | 0.0000622 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A056236 | PGDB_C019903 | PGDB_AS002246 | View |
| Dmax | - | = | 1.53 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A058153 | PGDB_C019903 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000622 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A060374 | PGDB_C019903 | PGDB_AS001381 | View |
| EC50 | - | = | 0.0000000056 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A067156 | PGDB_C019903 | PGDB_AS002126 | View |
| EC50 | - | = | 0.0000622 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A067844 | PGDB_C019903 | PGDB_AS001009 | View |
| Dmax | - | = | 8.75 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A068077 | PGDB_C019903 | PGDB_AS001280 | View |