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Cc1ccc(F)c(-n2nnnc2SCc2ccccc2F)c1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 8.63 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A008227 | PGDB_C019904 | PGDB_AS001280 | View | |
| Dmax | - | = | 1.65 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A012885 | PGDB_C019904 | PGDB_AS000546 | View | |
| Dmax | - | = | 2.47 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A014582 | PGDB_C019904 | PGDB_AS000856 | View | |
| EC50 | - | = | 0.0000729 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A024813 | PGDB_C019904 | PGDB_AS001381 | View | |
| EC50 | - | = | 0.0000000082 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A026229 | PGDB_C019904 | PGDB_AS000046 | View | |
| EC50 | - | = | 0.0000729 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A031796 | PGDB_C019904 | PGDB_AS002246 | View | |
| EC50 | - | = | 0.0000729 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A049569 | PGDB_C019904 | PGDB_AS001009 | View | |
| EC50 | - | = | 0.0000000027 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A056253 | PGDB_C019904 | PGDB_AS001078 | View | |
| EC50 | - | = | 0.0000000102 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A071857 | PGDB_C019904 | PGDB_AS002126 | View |