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CCOc1ccc(Br)cc1C1C2=C(CCCC2=O)N(CC(=O)O)C2=C1C(=O)CCC2| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000000054 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A014340 | PGDB_C019905 | PGDB_AS000046 | View | |
| Dmax | - | = | 8.52 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A020345 | PGDB_C019905 | PGDB_AS001280 | View | |
| EC50 | - | = | 0.0000436 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A032281 | PGDB_C019905 | PGDB_AS001381 | View | |
| Dmax | - | = | 1.87 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A036455 | PGDB_C019905 | PGDB_AS000546 | View | |
| EC50 | - | = | 0.0000000011 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A054681 | PGDB_C019905 | PGDB_AS001078 | View | |
| EC50 | - | = | 0.0000000052 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A057730 | PGDB_C019905 | PGDB_AS002126 | View | |
| EC50 | - | = | 0.0000436 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A058184 | PGDB_C019905 | PGDB_AS001009 | View | |
| Dmax | - | = | 2.3 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A061036 | PGDB_C019905 | PGDB_AS000856 | View | |
| EC50 | - | = | 0.0000436 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A065476 | PGDB_C019905 | PGDB_AS002246 | View |