Loading compound
Loading detail record from the SQLite release...
Loading detail record from the SQLite release...
CC1=C(C(=O)OCc2ccccc2)C(c2cn(-c3ccccc3)nc2-c2ccc(F)cc2)C(C(=O)OCc2ccccc2)=C(C)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000000034 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A009689 | PGDB_C019907 | PGDB_AS000046 | View | |
| EC50 | - | = | 0.0000342 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A011231 | PGDB_C019907 | PGDB_AS001381 | View | |
| Dmax | - | = | 8.34 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A038337 | PGDB_C019907 | PGDB_AS001280 | View | |
| EC50 | - | = | 0.0000000018 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A059144 | PGDB_C019907 | PGDB_AS002126 | View | |
| EC50 | - | = | 0.0000342 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A059728 | PGDB_C019907 | PGDB_AS001009 | View | |
| Dmax | - | = | 2.59 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A061490 | PGDB_C019907 | PGDB_AS000856 | View | |
| EC50 | - | = | 0.0000000004498 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A065134 | PGDB_C019907 | PGDB_AS001078 | View | |
| EC50 | - | = | 0.0000342 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A066422 | PGDB_C019907 | PGDB_AS002246 | View | |
| Dmax | - | = | 1.54 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A069122 | PGDB_C019907 | PGDB_AS000546 | View |