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Cc1cc(OCC(=O)Nc2ccc3oc(-c4ccccc4Br)nc3c2)cc(C)c1Cl| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000432 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A013932 | PGDB_C019908 | PGDB_AS002246 | View | |
| EC50 | - | = | 0.0001255 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A015960 | PGDB_C019908 | PGDB_AS002126 | View | |
| EC50 | - | = | 0.0000000206 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A018978 | PGDB_C019908 | PGDB_AS001078 | View | |
| Dmax | - | = | 0.32 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A023261 | PGDB_C019908 | PGDB_AS000546 | View | |
| EC50 | - | = | 0.0000000412 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A023960 | PGDB_C019908 | PGDB_AS000046 | View | |
| Dmax | - | = | 0.02 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A028257 | PGDB_C019908 | PGDB_AS000856 | View | |
| EC50 | - | = | 0.0000432 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A045889 | PGDB_C019908 | PGDB_AS001009 | View | |
| Dmax | - | = | 8.15 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A057552 | PGDB_C019908 | PGDB_AS001280 | View | |
| EC50 | - | = | 0.0000432 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A062405 | PGDB_C019908 | PGDB_AS001381 | View |