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CCSCCOC(=O)C1=C(C)NC2=C(C(=O)CC(c3ccccc3)C2)C1c1ccc(OC)cc1OC| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000414 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A023535 | PGDB_C019909 | PGDB_AS001009 | View | |
| EC50 | - | = | 0.0000000036 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A026403 | PGDB_C019909 | PGDB_AS000046 | View | |
| EC50 | - | = | 0.0000000044 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A036263 | PGDB_C019909 | PGDB_AS002126 | View | |
| Dmax | - | = | 2.61 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A052333 | PGDB_C019909 | PGDB_AS000856 | View | |
| Dmax | - | = | 7.92 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A055329 | PGDB_C019909 | PGDB_AS001280 | View | |
| EC50 | - | = | 0.0000414 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A059221 | PGDB_C019909 | PGDB_AS001381 | View | |
| EC50 | - | = | 0.0000000026 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A064183 | PGDB_C019909 | PGDB_AS001078 | View | |
| EC50 | - | = | 0.0000414 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A073362 | PGDB_C019909 | PGDB_AS002246 | View | |
| Dmax | - | = | 0.91 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A076859 | PGDB_C019909 | PGDB_AS000546 | View |