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Compound
PGDB_C019910
9 activity records1 related patents
2D structure
CCSCCOC(=O)C1=C(C)NC2=C(C(=O)CC(C)C2)C1c1ccc(Br)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000245 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A012380 | PGDB_C019910 | PGDB_AS002126 | View |
| EC50 | - | = | 0.0000544 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A018000 | PGDB_C019910 | PGDB_AS001009 | View |
| EC50 | - | = | 0.0000071 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A022838 | PGDB_C019910 | PGDB_AS000046 | View |
| Dmax | - | = | 0.86 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A023518 | PGDB_C019910 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000464 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A031004 | PGDB_C019910 | PGDB_AS001078 | View |
| Dmax | - | = | 0.21 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A041397 | PGDB_C019910 | PGDB_AS000856 | View |
| EC50 | - | = | 0.0000544 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A053858 | PGDB_C019910 | PGDB_AS002246 | View |
| Dmax | - | = | 7.86 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A062818 | PGDB_C019910 | PGDB_AS001280 | View |
| EC50 | - | = | 0.0000544 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A064890 | PGDB_C019910 | PGDB_AS001381 | View |