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Compound
PGDB_C019912
9 activity records1 related patents
2D structure
Cc1ccc2c(CC(=O)Nc3ccc(F)c(Cl)c3)nn(C)c(=O)c2c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 0.04 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A017522 | PGDB_C019912 | PGDB_AS000856 | View |
| Dmax | - | = | 7.32 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A017924 | PGDB_C019912 | PGDB_AS001280 | View |
| Dmax | - | = | -0.2468 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A020011 | PGDB_C019912 | PGDB_AS000546 | View |
| EC50 | - | = | 0.000085 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A030622 | PGDB_C019912 | PGDB_AS001381 | View |
| EC50 | - | = | 0.0000168 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A033087 | PGDB_C019912 | PGDB_AS001078 | View |
| EC50 | - | = | 0.0000006984 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A045017 | PGDB_C019912 | PGDB_AS000046 | View |
| EC50 | - | = | 0.000085 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A053634 | PGDB_C019912 | PGDB_AS001009 | View |
| EC50 | - | = | 0.000085 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A056489 | PGDB_C019912 | PGDB_AS002246 | View |
| EC50 | - | = | 0.0001129 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A077794 | PGDB_C019912 | PGDB_AS002126 | View |