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O=C(Nc1ccc2oc(-c3ccc4ccccc4c3)nc2c1)c1cccc(Cl)c1Cl| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 7.3 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A012254 | PGDB_C019913 | PGDB_AS001280 | View | |
| EC50 | - | = | 0.0000566 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A020187 | PGDB_C019913 | PGDB_AS002246 | View | |
| EC50 | - | = | 0.0000566 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A024341 | PGDB_C019913 | PGDB_AS001381 | View | |
| EC50 | - | = | 0.0000063 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A032376 | PGDB_C019913 | PGDB_AS001078 | View | |
| EC50 | - | = | 0.0000566 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A039399 | PGDB_C019913 | PGDB_AS001009 | View | |
| Dmax | - | = | 0.21 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A051710 | PGDB_C019913 | PGDB_AS000856 | View | |
| EC50 | - | = | 0.0000001355 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A054394 | PGDB_C019913 | PGDB_AS002126 | View | |
| EC50 | - | = | 0.0000000458 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A060201 | PGDB_C019913 | PGDB_AS000046 | View | |
| Dmax | - | = | -0.031 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A068416 | PGDB_C019913 | PGDB_AS000546 | View |