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Compound
PGDB_C019915
9 activity records1 related patents
2D structure
CC(C)c1ccc(Nc2nccn3c(-c4ccoc4)cnc23)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000127 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A007442 | PGDB_C019915 | PGDB_AS000046 | View |
| Dmax | - | = | 1.39 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A010792 | PGDB_C019915 | PGDB_AS000856 | View |
| EC50 | - | = | 0.0000139 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A024740 | PGDB_C019915 | PGDB_AS002126 | View |
| Dmax | - | = | -0.1894 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A031649 | PGDB_C019915 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0005615 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A036933 | PGDB_C019915 | PGDB_AS001078 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A039534 | PGDB_C019915 | PGDB_AS001381 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A051939 | PGDB_C019915 | PGDB_AS001009 | View |
| Dmax | - | = | 6.99 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A057543 | PGDB_C019915 | PGDB_AS001280 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A070362 | PGDB_C019915 | PGDB_AS002246 | View |