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Compound
PGDB_C019916
9 activity records1 related patents
2D structure
Cc1cccc(C(=O)N/C(=C/c2ccccc2)C(=O)Nc2c(C)n(C)n(-c3ccccc3)c2=O)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 0.11 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A011767 | PGDB_C019916 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000004957 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A015012 | PGDB_C019916 | PGDB_AS001078 | View |
| EC50 | - | = | 0.0000000401 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A016462 | PGDB_C019916 | PGDB_AS000046 | View |
| EC50 | - | = | 0.0000567 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A018118 | PGDB_C019916 | PGDB_AS002246 | View |
| Dmax | - | = | 6.91 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A022071 | PGDB_C019916 | PGDB_AS001280 | View |
| EC50 | - | = | 0.0000567 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A025777 | PGDB_C019916 | PGDB_AS001381 | View |
| EC50 | - | = | 0.0000006186 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A034471 | PGDB_C019916 | PGDB_AS002126 | View |
| EC50 | - | = | 0.0000567 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A037965 | PGDB_C019916 | PGDB_AS001009 | View |
| Dmax | - | = | 0.18 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A048581 | PGDB_C019916 | PGDB_AS000856 | View |