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Compound
PGDB_C019917
9 activity records1 related patents
2D structure
CC(NC(=O)c1cnc2ccccn12)c1ccc(F)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000000903 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A009207 | PGDB_C019917 | PGDB_AS000046 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A016188 | PGDB_C019917 | PGDB_AS002246 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A018740 | PGDB_C019917 | PGDB_AS001381 | View |
| EC50 | - | = | 0.0000002638 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A019752 | PGDB_C019917 | PGDB_AS001078 | View |
| Dmax | - | = | 6.66 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A040505 | PGDB_C019917 | PGDB_AS001280 | View |
| Dmax | - | = | 1.12 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A040969 | PGDB_C019917 | PGDB_AS000546 | View |
| EC50 | - | = | 0.000000011 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A065107 | PGDB_C019917 | PGDB_AS002126 | View |
| Dmax | - | = | 0.23 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A069953 | PGDB_C019917 | PGDB_AS000856 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A070320 | PGDB_C019917 | PGDB_AS001009 | View |