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Compound
PGDB_C019918
9 activity records1 related patents
2D structure
Cc1ccnc(N2CCC(C(=O)Nc3ccccc3Br)CC2)n1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A019690 | PGDB_C019918 | PGDB_AS001009 | View |
| Dmax | - | = | 6.46 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A035488 | PGDB_C019918 | PGDB_AS001280 | View |
| EC50 | - | = | 0.0000000024 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A043972 | PGDB_C019918 | PGDB_AS001078 | View |
| Dmax | - | = | 0.05 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A050195 | PGDB_C019918 | PGDB_AS000856 | View |
| EC50 | - | = | 0.0000000033 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A056291 | PGDB_C019918 | PGDB_AS002126 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A062532 | PGDB_C019918 | PGDB_AS002246 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A064567 | PGDB_C019918 | PGDB_AS001381 | View |
| Dmax | - | = | 0.25 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A068490 | PGDB_C019918 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000000482 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A071844 | PGDB_C019918 | PGDB_AS000046 | View |