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CCC(c1nnnn1CCC(C)C)N1CCN(C(=O)c2cc(C)co2)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 0.18 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A009592 | PGDB_C019919 | PGDB_AS000856 | View | |
| EC50 | - | = | 0.0000023 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A010864 | PGDB_C019919 | PGDB_AS002126 | View | |
| EC50 | - | = | 0.0002347 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A032289 | PGDB_C019919 | PGDB_AS001078 | View | |
| Dmax | - | = | 0.87 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A042872 | PGDB_C019919 | PGDB_AS000546 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A045409 | PGDB_C019919 | PGDB_AS001381 | View | |
| Dmax | - | = | 6.45 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A045677 | PGDB_C019919 | PGDB_AS001280 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A050924 | PGDB_C019919 | PGDB_AS002246 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A070387 | PGDB_C019919 | PGDB_AS001009 | View | |
| EC50 | - | = | 0.000024 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A077749 | PGDB_C019919 | PGDB_AS000046 | View |