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Compound
PGDB_C019920
9 activity records1 related patents
2D structure
C=C1c2cnn(-c3ccccc3)c2N=NN1Cc1cccnc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A015845 | PGDB_C019920 | PGDB_AS002246 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A019348 | PGDB_C019920 | PGDB_AS001381 | View |
| Dmax | - | = | 2.7 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A019973 | PGDB_C019920 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A025685 | PGDB_C019920 | PGDB_AS001009 | View |
| EC50 | - | = | 0.0000119 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A025792 | PGDB_C019920 | PGDB_AS002126 | View |
| EC50 | - | = | 0.000000009 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A032527 | PGDB_C019920 | PGDB_AS000046 | View |
| Dmax | - | = | 0.12 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A037384 | PGDB_C019920 | PGDB_AS000856 | View |
| EC50 | - | = | 0.0001102 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A052874 | PGDB_C019920 | PGDB_AS001078 | View |
| Dmax | - | = | 6.4 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A061168 | PGDB_C019920 | PGDB_AS001280 | View |