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O=C(NCCCN1CCc2ccccc2C1)Nc1ccc(Br)cc1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 0.28 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A011444 | PGDB_C019921 | PGDB_AS000856 | View | |
| Dmax | - | = | 6.18 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A019327 | PGDB_C019921 | PGDB_AS001280 | View | |
| Dmax | - | = | -0.0757 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A022140 | PGDB_C019921 | PGDB_AS000546 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A032674 | PGDB_C019921 | PGDB_AS001009 | View | |
| EC50 | - | = | 0.0000000093 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A037286 | PGDB_C019921 | PGDB_AS001078 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A046688 | PGDB_C019921 | PGDB_AS002246 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A058103 | PGDB_C019921 | PGDB_AS001381 | View | |
| EC50 | - | = | 0.0000002554 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A061905 | PGDB_C019921 | PGDB_AS002126 | View | |
| EC50 | - | = | 0.0000002554 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A074996 | PGDB_C019921 | PGDB_AS000046 | View |