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Compound
PGDB_C021157
9 activity records1 related patents
2D structure
CCCOc1ccc(C2C(C(=O)OC)=CN(CCOC)C=C2C(=O)OC(F)(F)F)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A010011 | PGDB_C021157 | PGDB_AS001381 | View |
| EC50 | - | = | 0.000019 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A025061 | PGDB_C021157 | PGDB_AS002126 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A025622 | PGDB_C021157 | PGDB_AS002246 | View |
| Dmax | - | = | 0.31 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A049570 | PGDB_C021157 | PGDB_AS000856 | View |
| Dmax | - | = | 5.19 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A062719 | PGDB_C021157 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000219 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A063883 | PGDB_C021157 | PGDB_AS000046 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A063959 | PGDB_C021157 | PGDB_AS001009 | View |
| Dmax | - | = | 10.71 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A070204 | PGDB_C021157 | PGDB_AS001280 | View |
| EC50 | - | = | 0.0000000000076 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A072326 | PGDB_C021157 | PGDB_AS001078 | View |