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Compound
PGDB_C021158
9 activity records1 related patents
2D structure
CCN(Cc1ccccc1)C(=O)c1cc2c(=O)n3ccc(C)c(C)c3nc2n1CCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000041 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A014225 | PGDB_C021158 | PGDB_AS002126 | View |
| Dmax | - | = | 1.56 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A020666 | PGDB_C021158 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A020707 | PGDB_C021158 | PGDB_AS001009 | View |
| Dmax | - | = | 0.79 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A035648 | PGDB_C021158 | PGDB_AS000856 | View |
| Dmax | - | = | 8.52 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A051318 | PGDB_C021158 | PGDB_AS001280 | View |
| EC50 | - | = | 0.0000001442 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A052180 | PGDB_C021158 | PGDB_AS001078 | View |
| EC50 | - | = | 0.0000215 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A054927 | PGDB_C021158 | PGDB_AS000046 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A072533 | PGDB_C021158 | PGDB_AS001381 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A072980 | PGDB_C021158 | PGDB_AS002246 | View |