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SIMM · NJU
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·
SIMM · NJU
Target
RBM39
661 activity records
561 compounds
6 patents
Target summary
Target ID
PGDB_T000086
Name
RBM39
Gene symbol
RBM39
Protein name
RNA-binding protein 39
UniProt ID
Q14498
Role
degradation_target | neo_substrate | primary_target
Compounds
561
Activity records
661
Assays
10
Patents
6
Activity compounds and values
Activity records
661 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
500-1000
nM
-
—
RBM39
-
HCT116
WO2025189015A1
PGDB_A007043
PGDB_C027673
PGDB_AS000963
View
EC50
-
=
179.6
nM
-
—
RBM39
DCAF15
-
EP4634155A1
PGDB_A007065
PGDB_C007837
PGDB_AS001059
View
EC50
-
=
353.8
nM
-
—
RBM39
DCAF15
-
EP4573088A1
PGDB_A007098
PGDB_C007602
PGDB_AS000315
View
EC50
-
<=
100
uM
-
—
RBM39
DCAF15
-
WO2023059899A1
PGDB_A007124
PGDB_C010022
PGDB_AS001283
View
EC50
-
<
10
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A007146
PGDB_C009790
PGDB_AS000136
View
EC50
-
=
4425.9
nM
-
—
RBM39
DCAF15
-
EP4634155A1
PGDB_A007208
PGDB_C007873
PGDB_AS001059
View
EC50
-
=
4190.8
nM
-
—
RBM39
DCAF15
-
EP4573088A1
PGDB_A007935
PGDB_C007604
PGDB_AS000315
View
EC50
-
=
0.0026
uM
-
—
RBM39
DCAF15
-
AR127239A1
PGDB_A008133
PGDB_C005605
PGDB_AS002536
View
EC50
-
=
0.0031
uM
-
—
RBM39
DCAF15
-
AR127239A1
PGDB_A008138
PGDB_C005555
PGDB_AS002536
View
EC50
-
>
100
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A008240
PGDB_C009647
PGDB_AS000136
View
EC50
-
<=
10
uM
-
—
RBM39
DCAF15
-
WO2023059899A1
PGDB_A008442
PGDB_C010016
PGDB_AS001283
View
EC50
-
=
3262.1
nM
-
—
RBM39
DCAF15
-
EP4573088A1
PGDB_A008563
PGDB_C007666
PGDB_AS000315
View
IC50
-
=
500-1000
nM
-
—
RBM39
-
HCT116
WO2025189015A1
PGDB_A008800
PGDB_C027671
PGDB_AS000963
View
EC50
-
<
10
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A008923
PGDB_C009677
PGDB_AS000136
View
EC50
-
=
0.0011
uM
-
—
RBM39
DCAF15
-
AR127239A1
PGDB_A008990
PGDB_C005599
PGDB_AS002536
View
IC50
-
=
1.791
uM
-
—
RBM39
-
HCT116
AR127239A1
PGDB_A009052
PGDB_C005633
PGDB_AS002257
View
EC50
-
=
0.0007
uM
-
—
RBM39
DCAF15
-
AR127239A1
PGDB_A009083
PGDB_C005627
PGDB_AS002536
View
EC50
-
<=
1
uM
-
—
RBM39
DCAF15
-
WO2023059899A1
PGDB_A009262
PGDB_C010009
PGDB_AS001283
View
EC50
-
<
10
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A009492
PGDB_C009646
PGDB_AS000136
View
EC50
-
=
88.7
nM
-
—
RBM39
DCAF15
-
EP4634155A1
PGDB_A009515
PGDB_C007827
PGDB_AS001059
View