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SIMM · NJU
Assay
PGDB_AS000368
System: biochemical
Target: CRBN
Assay context summary
Assay context
50 activity records
Assay family
binding
System
biochemical
Readout
Kd
Target
CRBN
E3
CRBN
Activity compounds and values
Activity records
50 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Kd
-
=
0.13
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A007345
PGDB_C007983
PGDB_AS000368
View
Kd
-
=
0.15
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A009850
PGDB_C008016
PGDB_AS000368
View
Kd
-
=
0.35
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A011604
PGDB_C007996
PGDB_AS000368
View
Kd
-
=
0.074
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A012659
PGDB_C007997
PGDB_AS000368
View
Kd
-
=
0.04
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A014867
PGDB_C007988
PGDB_AS000368
View
Kd
-
=
0.18
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A015131
PGDB_C008012
PGDB_AS000368
View
Kd
-
=
0.23
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A016014
PGDB_C008014
PGDB_AS000368
View
Kd
-
=
0.84
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A019382
PGDB_C007995
PGDB_AS000368
View
Kd
-
=
0.13
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A020393
PGDB_C008015
PGDB_AS000368
View
Kd
-
=
0.31
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A021771
PGDB_C007992
PGDB_AS000368
View
Kd
-
=
0.045
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A022452
PGDB_C008001
PGDB_AS000368
View
Kd
-
=
0.26
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A023243
PGDB_C007971
PGDB_AS000368
View
Kd
-
=
0.73
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A027511
PGDB_C007972
PGDB_AS000368
View
Kd
-
=
0.21
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A029894
PGDB_C007987
PGDB_AS000368
View
Kd
-
=
0.34
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A029989
PGDB_C008004
PGDB_AS000368
View
Kd
-
=
0.2
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A031969
PGDB_C007998
PGDB_AS000368
View
Kd
-
=
0.44
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A032178
PGDB_C007985
PGDB_AS000368
View
Kd
-
=
0.23
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A035734
PGDB_C008006
PGDB_AS000368
View
Kd
-
=
0.35
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A039105
PGDB_C007986
PGDB_AS000368
View
Kd
-
=
0.36
uM
-
—
CRBN
CRBN
-
WO2025043225
PGDB_A043587
PGDB_C008002
PGDB_AS000368
View