Assay context summary

Assay context

18 activity records
Activity compounds and values

Activity records

18 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C008162
IC50-=61.4nM-GSPT1-NCI-H1155IL323841APGDB_A007532PGDB_C008162PGDB_AS000925View
2D structure for PGDB_C008153
IC50-=38.4nM-GSPT1-NCI-H1155IL323841APGDB_A018837PGDB_C008153PGDB_AS000925View
2D structure for PGDB_C008155
IC50-=100.8nM-GSPT1-NCI-H1155IL323841APGDB_A019205PGDB_C008155PGDB_AS000925View
2D structure for PGDB_C008164
IC50-=34.3nM-GSPT1-NCI-H1155IL323841APGDB_A021956PGDB_C008164PGDB_AS000925View
2D structure for PGDB_C008168
IC50-=36nM-GSPT1-NCI-H1155IL323841APGDB_A024670PGDB_C008168PGDB_AS000925View
2D structure for PGDB_C008157
IC50-=24.1nM-GSPT1-NCI-H1155IL323841APGDB_A025100PGDB_C008157PGDB_AS000925View
2D structure for PGDB_C008161
IC50-=53.1nM-GSPT1-NCI-H1155IL323841APGDB_A028843PGDB_C008161PGDB_AS000925View
2D structure for PGDB_C001361
IC50-=129nM-GSPT1-NCI-H1155IL323841APGDB_A029785PGDB_C001361PGDB_AS000925View
2D structure for PGDB_C008166
IC50-=15.7nM-GSPT1-NCI-H1155IL323841APGDB_A032825PGDB_C008166PGDB_AS000925View
2D structure for PGDB_C019545
IC50-=114nM-GSPT1-NCI-H1155IL323841APGDB_A035998PGDB_C019545PGDB_AS000925View
2D structure for PGDB_C008163
IC50-=59.4nM-GSPT1-NCI-H1155IL323841APGDB_A045045PGDB_C008163PGDB_AS000925View
2D structure for PGDB_C008154
IC50-=148nM-GSPT1-NCI-H1155IL323841APGDB_A052138PGDB_C008154PGDB_AS000925View
2D structure for PGDB_C008151
IC50-=26.7nM-GSPT1-NCI-H1155IL323841APGDB_A053229PGDB_C008151PGDB_AS000925View
2D structure for PGDB_C008150
IC50-=43.1nM-GSPT1-NCI-H1155IL323841APGDB_A056483PGDB_C008150PGDB_AS000925View
2D structure for PGDB_C008149
IC50-=44.6nM-GSPT1-NCI-H1155IL323841APGDB_A064189PGDB_C008149PGDB_AS000925View
2D structure for PGDB_C008165
IC50-=60.2nM-GSPT1-NCI-H1155IL323841APGDB_A065661PGDB_C008165PGDB_AS000925View
2D structure for PGDB_C008167
IC50-=30.1nM-GSPT1-NCI-H1155IL323841APGDB_A065793PGDB_C008167PGDB_AS000925View
2D structure for PGDB_C008152
IC50-=34.5nM-GSPT1-NCI-H1155IL323841APGDB_A070685PGDB_C008152PGDB_AS000925View