Assay context summary

Assay context

22 activity records
Activity compounds and values

Activity records

22 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000360
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A015573PGDB_C000360PGDB_AS000935View
2D structure for PGDB_C000363
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A017750PGDB_C000363PGDB_AS000935View
2D structure for PGDB_C000359
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A019319PGDB_C000359PGDB_AS000935View
2D structure for PGDB_C000370
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A019479PGDB_C000370PGDB_AS000935View
2D structure for PGDB_C000376
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A022109PGDB_C000376PGDB_AS000935View
2D structure for PGDB_C000375
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A030296PGDB_C000375PGDB_AS000935View
2D structure for PGDB_C000377
IC50-=1000-2000nM-BRD4/GSPT1-NB4CN117756818APGDB_A034049PGDB_C000377PGDB_AS000935View
2D structure for PGDB_C000373
IC50-=4.1nM-BRD4/GSPT1-NB4CN117756818APGDB_A034260PGDB_C000373PGDB_AS000935View
2D structure for PGDB_C000379
IC50-=100-1000nM-BRD4/GSPT1-NB4CN117756818APGDB_A034720PGDB_C000379PGDB_AS000935View
2D structure for PGDB_C000362
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A044540PGDB_C000362PGDB_AS000935View
2D structure for PGDB_C000372
IC50-=7.8nM-BRD4/GSPT1-NB4CN117756818APGDB_A051425PGDB_C000372PGDB_AS000935View
2D structure for PGDB_C000369
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A052795PGDB_C000369PGDB_AS000935View
2D structure for PGDB_C000367
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A054465PGDB_C000367PGDB_AS000935View
2D structure for PGDB_C000368
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A056022PGDB_C000368PGDB_AS000935View
2D structure for PGDB_C000365
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A056679PGDB_C000365PGDB_AS000935View
2D structure for PGDB_C000364
IC50-=13.4nM-BRD4/GSPT1-NB4CN117756818APGDB_A058062PGDB_C000364PGDB_AS000935View
2D structure for PGDB_C000378
IC50-=100-1000nM-BRD4/GSPT1-NB4CN117756818APGDB_A058844PGDB_C000378PGDB_AS000935View
2D structure for PGDB_C000371
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A065117PGDB_C000371PGDB_AS000935View
2D structure for PGDB_C000366
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A067174PGDB_C000366PGDB_AS000935View
2D structure for PGDB_C000361
IC50-<100nM-BRD4/GSPT1-NB4CN117756818APGDB_A071114PGDB_C000361PGDB_AS000935View