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SIMM · NJU
Assay
PGDB_AS000935
System: cell_based
Target: BRD4
Cell line: NB4
Assay context summary
Assay context
22 activity records
Assay family
viability
System
cell_based
Readout
IC50
Target
BRD4
E3
Not specified
Cell line
NB4
Activity compounds and values
Activity records
22 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A015573
PGDB_C000360
PGDB_AS000935
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A017750
PGDB_C000363
PGDB_AS000935
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A019319
PGDB_C000359
PGDB_AS000935
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A019479
PGDB_C000370
PGDB_AS000935
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A022109
PGDB_C000376
PGDB_AS000935
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A030296
PGDB_C000375
PGDB_AS000935
View
IC50
-
=
1000-2000
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A034049
PGDB_C000377
PGDB_AS000935
View
IC50
-
=
4.1
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A034260
PGDB_C000373
PGDB_AS000935
View
IC50
-
=
100-1000
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A034720
PGDB_C000379
PGDB_AS000935
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A044540
PGDB_C000362
PGDB_AS000935
View
IC50
-
=
7.8
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A051425
PGDB_C000372
PGDB_AS000935
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A052795
PGDB_C000369
PGDB_AS000935
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A054465
PGDB_C000367
PGDB_AS000935
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A056022
PGDB_C000368
PGDB_AS000935
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A056679
PGDB_C000365
PGDB_AS000935
View
IC50
-
=
13.4
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A058062
PGDB_C000364
PGDB_AS000935
View
IC50
-
=
100-1000
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A058844
PGDB_C000378
PGDB_AS000935
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A065117
PGDB_C000371
PGDB_AS000935
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A067174
PGDB_C000366
PGDB_AS000935
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
NB4
CN117756818A
PGDB_A071114
PGDB_C000361
PGDB_AS000935
View