Assay
PGDB_AS001216
System: cell_basedTarget: CRBN | DDB1Cell line: HEK293
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Kd | - | = | 7.3 | nM | - | — | CRBN | CRBN | HEK293 | IL323841A | PGDB_A010767 | PGDB_C008152 | PGDB_AS001216 | View | |
| Kd | - | = | 7.9 | nM | - | — | CRBN | CRBN | HEK293 | IL323841A | PGDB_A017003 | PGDB_C008153 | PGDB_AS001216 | View | |
| Kd | - | = | 28 | nM | - | — | CRBN | CRBN | HEK293 | IL323841A | PGDB_A020755 | PGDB_C008149 | PGDB_AS001216 | View | |
| Kd | - | = | 6.2 | nM | - | — | CRBN | CRBN | HEK293 | IL323841A | PGDB_A027716 | PGDB_C008150 | PGDB_AS001216 | View | |
| Kd | - | = | 3.5 | nM | - | — | CRBN | CRBN | HEK293 | IL323841A | PGDB_A047395 | PGDB_C008151 | PGDB_AS001216 | View | |
| Kd | - | = | 9.9 | nM | - | — | CRBN | CRBN | HEK293 | IL323841A | PGDB_A050246 | PGDB_C019545 | PGDB_AS001216 | View | |
| Kd | - | = | 8.6 | nM | - | — | CRBN | CRBN | HEK293 | IL323841A | PGDB_A061475 | PGDB_C008154 | PGDB_AS001216 | View | |
| Kd | - | = | 6 | nM | - | — | CRBN | CRBN | HEK293 | IL323841A | PGDB_A063862 | PGDB_C001361 | PGDB_AS001216 | View | |
| Kd | - | = | 7.2 | nM | - | — | CRBN | CRBN | HEK293 | IL323841A | PGDB_A076839 | PGDB_C008155 | PGDB_AS001216 | View |