Assay
PGDB_AS001647
System: cell_based
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | >= | 0 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A007177 | PGDB_C019406 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 20 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A007216 | PGDB_C019255 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 0 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A007246 | PGDB_C019434 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 0 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A007264 | PGDB_C019424 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 20 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A007577 | PGDB_C019307 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 20 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A007693 | PGDB_C019382 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 0 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A007992 | PGDB_C019300 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 0 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A008038 | PGDB_C019507 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 20 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A008202 | PGDB_C019403 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 20 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A008477 | PGDB_C019220 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 0 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A008667 | PGDB_C019419 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 20 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A008792 | PGDB_C019277 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 20 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A009140 | PGDB_C019265 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 20 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A009374 | PGDB_C019186 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 20 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A009380 | PGDB_C019340 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 20 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A009805 | PGDB_C019189 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 0 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A009946 | PGDB_C019449 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 0 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A009971 | PGDB_C019182 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 20 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A010669 | PGDB_C019386 | PGDB_AS001647 | View | |
| % Degradation | - | >= | 0 | % | Concentration series: 500 nM, 50 nM | 24 h | CSNK1A1 | - | - | WO2025016359A1 | PGDB_A010759 | PGDB_C019395 | PGDB_AS001647 | View |