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SIMM · NJU
Assay
PGDB_AS002081
System: cell_based
Target: BRD4
Cell line: Oci-AML3
Assay context summary
Assay context
22 activity records
Assay family
viability
System
cell_based
Readout
IC50
Target
BRD4
E3
Not specified
Cell line
Oci-AML3
Activity compounds and values
Activity records
22 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
100-1000
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A012063
PGDB_C000361
PGDB_AS002081
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A012688
PGDB_C000365
PGDB_AS002081
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A013614
PGDB_C000366
PGDB_AS002081
View
IC50
-
=
100-1000
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A015700
PGDB_C000360
PGDB_AS002081
View
IC50
-
>
2000
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A019468
PGDB_C000379
PGDB_AS002081
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A024602
PGDB_C000367
PGDB_AS002081
View
IC50
-
=
100-1000
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A025568
PGDB_C000359
PGDB_AS002081
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A025765
PGDB_C000369
PGDB_AS002081
View
IC50
-
>
2000
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A032790
PGDB_C000377
PGDB_AS002081
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A034467
PGDB_C000368
PGDB_AS002081
View
IC50
-
=
12
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A037694
PGDB_C000373
PGDB_AS002081
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A037969
PGDB_C000372
PGDB_AS002081
View
IC50
-
=
100-1000
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A046534
PGDB_C000362
PGDB_AS002081
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A052862
PGDB_C000376
PGDB_AS002081
View
IC50
-
=
17.57
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A058688
PGDB_C000374
PGDB_AS002081
View
IC50
-
>
2000
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A059584
PGDB_C000378
PGDB_AS002081
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A060687
PGDB_C000370
PGDB_AS002081
View
IC50
-
>
2000
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A065183
PGDB_C000059
PGDB_AS002081
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A071135
PGDB_C000371
PGDB_AS002081
View
IC50
-
<
100
nM
-
—
BRD4/GSPT1
-
Oci-AML3
CN117756818A
PGDB_A072434
PGDB_C000375
PGDB_AS002081
View