Assay context summary

Assay context

22 activity records
Activity compounds and values

Activity records

22 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000361
IC50-=100-1000nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A012063PGDB_C000361PGDB_AS002081View
2D structure for PGDB_C000365
IC50-<100nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A012688PGDB_C000365PGDB_AS002081View
2D structure for PGDB_C000366
IC50-<100nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A013614PGDB_C000366PGDB_AS002081View
2D structure for PGDB_C000360
IC50-=100-1000nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A015700PGDB_C000360PGDB_AS002081View
2D structure for PGDB_C000379
IC50->2000nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A019468PGDB_C000379PGDB_AS002081View
2D structure for PGDB_C000367
IC50-<100nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A024602PGDB_C000367PGDB_AS002081View
2D structure for PGDB_C000359
IC50-=100-1000nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A025568PGDB_C000359PGDB_AS002081View
2D structure for PGDB_C000369
IC50-<100nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A025765PGDB_C000369PGDB_AS002081View
2D structure for PGDB_C000377
IC50->2000nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A032790PGDB_C000377PGDB_AS002081View
2D structure for PGDB_C000368
IC50-<100nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A034467PGDB_C000368PGDB_AS002081View
2D structure for PGDB_C000373
IC50-=12nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A037694PGDB_C000373PGDB_AS002081View
2D structure for PGDB_C000372
IC50-<100nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A037969PGDB_C000372PGDB_AS002081View
2D structure for PGDB_C000362
IC50-=100-1000nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A046534PGDB_C000362PGDB_AS002081View
2D structure for PGDB_C000376
IC50-<100nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A052862PGDB_C000376PGDB_AS002081View
2D structure for PGDB_C000374
IC50-=17.57nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A058688PGDB_C000374PGDB_AS002081View
2D structure for PGDB_C000378
IC50->2000nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A059584PGDB_C000378PGDB_AS002081View
2D structure for PGDB_C000370
IC50-<100nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A060687PGDB_C000370PGDB_AS002081View
2D structure for PGDB_C000059
IC50->2000nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A065183PGDB_C000059PGDB_AS002081View
2D structure for PGDB_C000371
IC50-<100nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A071135PGDB_C000371PGDB_AS002081View
2D structure for PGDB_C000375
IC50-<100nM-BRD4/GSPT1-Oci-AML3CN117756818APGDB_A072434PGDB_C000375PGDB_AS002081View