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SIMM · NJU
Assay
PGDB_AS002240
System: cell_based
Target: CDK2
Cell line: HEK293
Assay context summary
Assay context
15 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
CDK2
E3
Not specified
Cell line
HEK293
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
15 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
50
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A011245
PGDB_C008030
PGDB_AS002240
View
Dmax
-
=
40
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A013022
PGDB_C008029
PGDB_AS002240
View
Dmax
-
=
31
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A013328
PGDB_C008031
PGDB_AS002240
View
Dmax
-
=
42
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A020777
PGDB_C008033
PGDB_AS002240
View
Dmax
-
=
40
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A022383
PGDB_C008022
PGDB_AS002240
View
Dmax
-
=
50
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A027759
PGDB_C008021
PGDB_AS002240
View
Dmax
-
=
34
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A041454
PGDB_C008027
PGDB_AS002240
View
Dmax
-
=
33
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A044936
PGDB_C008024
PGDB_AS002240
View
Dmax
-
=
22
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A046930
PGDB_C008034
PGDB_AS002240
View
Dmax
-
=
38
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A053518
PGDB_C008026
PGDB_AS002240
View
Dmax
-
=
24
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A055285
PGDB_C008020
PGDB_AS002240
View
Dmax
-
=
38
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A062877
PGDB_C008025
PGDB_AS002240
View
Dmax
-
=
52
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A068451
PGDB_C008023
PGDB_AS002240
View
Dmax
-
=
41
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A070384
PGDB_C008028
PGDB_AS002240
View
Dmax
-
=
28
%
10 uM
18 h
CDK2
-
HEK293
WO2025043225
PGDB_A071993
PGDB_C008032
PGDB_AS002240
View