Assay

PGDB_AS002339

System: cell_basedTarget: GSPT1Cell line: HEK293
Assay context summary

Assay context

10 activity records
Assay family% Degradation
Systemcell_based
ReadoutDmax
TargetGSPT1
E3Not specified
Cell lineHEK293
OrganismHomo sapiens
Technologyluminescence
Detection targetprotein_degradation
Activity compounds and values

Activity records

10 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C001468
Dmax-=93.1%Concentration series: 1 uM24 hGSPT1-HEK293CN118852145APGDB_A016560PGDB_C001468PGDB_AS002339View
2D structure for PGDB_C001465
Dmax-=93.8%Concentration series: 1 uM24 hGSPT1-HEK293CN118852145APGDB_A021184PGDB_C001465PGDB_AS002339View
2D structure for PGDB_C001466
Dmax-=93.24%Concentration series: 1 uM24 hGSPT1-HEK293CN118852145APGDB_A022137PGDB_C001466PGDB_AS002339View
2D structure for PGDB_C001470
Dmax-=93.56%Concentration series: 1 uM24 hGSPT1-HEK293CN118852145APGDB_A024704PGDB_C001470PGDB_AS002339View
2D structure for PGDB_C001475
Dmax-=89.86%Concentration series: 1 uM24 hGSPT1-HEK293CN118852145APGDB_A025473PGDB_C001475PGDB_AS002339View
2D structure for PGDB_C001474
Dmax-=92.09%Concentration series: 1 uM24 hGSPT1-HEK293CN118852145APGDB_A027256PGDB_C001474PGDB_AS002339View
2D structure for PGDB_C001471
Dmax-=91.05%Concentration series: 1 uM24 hGSPT1-HEK293CN118852145APGDB_A031982PGDB_C001471PGDB_AS002339View
2D structure for PGDB_C001472
Dmax-=7.33%Concentration series: 1 uM24 hGSPT1-HEK293CN118852145APGDB_A035938PGDB_C001472PGDB_AS002339View
2D structure for PGDB_C001479
Dmax-=86.63%Concentration series: 1 uM24 hGSPT1-HEK293CN118852145APGDB_A063990PGDB_C001479PGDB_AS002339View
2D structure for PGDB_C001478
Dmax-=92.89%Concentration series: 1 uM24 hGSPT1-HEK293CN118852145APGDB_A064526PGDB_C001478PGDB_AS002339View
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