Assay

PGDB_AS002388

System: biochemicalTarget: CRBN | DDB1
Assay context summary

Assay context

17 activity records
Assay familybinding
Systembiochemical
ReadoutKi
TargetCRBN | DDB1
E3CRBN | DDB1
Technologyfluorescence
Activity compounds and values

Activity records

17 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C008998
Ki-=3.9uM-—CRBNCRBN-US12110292B2PGDB_A014004PGDB_C008998PGDB_AS002388View
2D structure for PGDB_C009000
Ki-=0.44uM-—CRBNCRBN-US12110292B2PGDB_A020041PGDB_C009000PGDB_AS002388View
2D structure for PGDB_C009001
Ki-=4.3uM-—CRBNCRBN-US12110292B2PGDB_A021458PGDB_C009001PGDB_AS002388View
2D structure for PGDB_C008993
Ki-=6.5uM-—CRBNCRBN-US12110292B2PGDB_A023556PGDB_C008993PGDB_AS002388View
2D structure for PGDB_C008992
Ki-=12.2uM-—CRBNCRBN-US12110292B2PGDB_A029078PGDB_C008992PGDB_AS002388View
2D structure for PGDB_C008995
Ki-=6.3uM-—CRBNCRBN-US12110292B2PGDB_A031464PGDB_C008995PGDB_AS002388View
2D structure for PGDB_C009002
Ki-=0.13uM-—CRBNCRBN-US12110292B2PGDB_A034262PGDB_C009002PGDB_AS002388View
2D structure for PGDB_C009003
Ki-=0.97uM-—CRBNCRBN-US12110292B2PGDB_A044325PGDB_C009003PGDB_AS002388View
2D structure for PGDB_C008988
Ki-=8.5uM-—CRBNCRBN-US12110292B2PGDB_A053432PGDB_C008988PGDB_AS002388View
2D structure for PGDB_C019024
Ki-=1.49uM-—CRBNCRBN-US12110292B2PGDB_A055171PGDB_C019024PGDB_AS002388View
2D structure for PGDB_C008990
Ki-=13.6uM-—CRBNCRBN-US12110292B2PGDB_A056754PGDB_C008990PGDB_AS002388View
2D structure for PGDB_C008997
Ki-=4.2uM-—CRBNCRBN-US12110292B2PGDB_A056796PGDB_C008997PGDB_AS002388View
2D structure for PGDB_C008999
Ki-=8.3uM-—CRBNCRBN-US12110292B2PGDB_A061296PGDB_C008999PGDB_AS002388View
2D structure for PGDB_C008994
Ki-=11.1uM-—CRBNCRBN-US12110292B2PGDB_A062433PGDB_C008994PGDB_AS002388View
2D structure for PGDB_C008996
Ki-=5.4uM-—CRBNCRBN-US12110292B2PGDB_A067401PGDB_C008996PGDB_AS002388View
2D structure for PGDB_C008989
Ki-=13.6uM-—CRBNCRBN-US12110292B2PGDB_A067899PGDB_C008989PGDB_AS002388View
2D structure for PGDB_C008991
Ki-=2.4uM-—CRBNCRBN-US12110292B2PGDB_A072513PGDB_C008991PGDB_AS002388View
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