Assay

PGDB_AS002405

System: cell_basedTarget: CDK2Cell line: HEK293
Assay context summary

Assay context

15 activity records
Assay family% Degradation
Systemcell_based
ReadoutIC50
TargetCDK2
E3Not specified
Cell lineHEK293
Technologyluminescence
Activity compounds and values

Activity records

15 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C008027
IC50-=0.22uM-—CDK2-HEK293WO2025043225PGDB_A014664PGDB_C008027PGDB_AS002405View
2D structure for PGDB_C008029
IC50-=0.032uM-—CDK2-HEK293WO2025043225PGDB_A016200PGDB_C008029PGDB_AS002405View
2D structure for PGDB_C008026
IC50-=0.2uM-—CDK2-HEK293WO2025043225PGDB_A021095PGDB_C008026PGDB_AS002405View
2D structure for PGDB_C008031
IC50-=0.99uM-—CDK2-HEK293WO2025043225PGDB_A023516PGDB_C008031PGDB_AS002405View
2D structure for PGDB_C008025
IC50-=0.083uM-—CDK2-HEK293WO2025043225PGDB_A026486PGDB_C008025PGDB_AS002405View
2D structure for PGDB_C008024
IC50-=0.24uM-—CDK2-HEK293WO2025043225PGDB_A027246PGDB_C008024PGDB_AS002405View
2D structure for PGDB_C008023
IC50-=0.066uM-—CDK2-HEK293WO2025043225PGDB_A028241PGDB_C008023PGDB_AS002405View
2D structure for PGDB_C008020
IC50-=0.19uM-—CDK2-HEK293WO2025043225PGDB_A030823PGDB_C008020PGDB_AS002405View
2D structure for PGDB_C008022
IC50-=0.044uM-—CDK2-HEK293WO2025043225PGDB_A031402PGDB_C008022PGDB_AS002405View
2D structure for PGDB_C008032
IC50-=0.18uM-—CDK2-HEK293WO2025043225PGDB_A033760PGDB_C008032PGDB_AS002405View
2D structure for PGDB_C008034
IC50-=0.31uM-—CDK2-HEK293WO2025043225PGDB_A041189PGDB_C008034PGDB_AS002405View
2D structure for PGDB_C008021
IC50-=0.054uM-—CDK2-HEK293WO2025043225PGDB_A042150PGDB_C008021PGDB_AS002405View
2D structure for PGDB_C008030
IC50-=0.091uM-—CDK2-HEK293WO2025043225PGDB_A047008PGDB_C008030PGDB_AS002405View
2D structure for PGDB_C008033
IC50-=0.13uM-—CDK2-HEK293WO2025043225PGDB_A058087PGDB_C008033PGDB_AS002405View
2D structure for PGDB_C008028
IC50-=0.092uM-—CDK2-HEK293WO2025043225PGDB_A077583PGDB_C008028PGDB_AS002405View
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