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SIMM · NJU
Assay
PGDB_AS002511
System: cell_based
Target: GSPT1
Cell line: HEK293
Assay context summary
Assay context
50 activity records
Assay family
% Degradation
System
cell_based
Readout
IC50
Target
GSPT1
E3
Not specified
Cell line
HEK293
Technology
luminescence
Activity compounds and values
Activity records
50 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A012079
PGDB_C007974
PGDB_AS002511
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A012357
PGDB_C008000
PGDB_AS002511
View
IC50
-
=
1
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A015244
PGDB_C008018
PGDB_AS002511
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A017033
PGDB_C007979
PGDB_AS002511
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A017889
PGDB_C007971
PGDB_AS002511
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A021434
PGDB_C007995
PGDB_AS002511
View
IC50
-
=
1
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A023423
PGDB_C008009
PGDB_AS002511
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A024580
PGDB_C007981
PGDB_AS002511
View
IC50
-
=
1
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A027118
PGDB_C008015
PGDB_AS002511
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A027717
PGDB_C007982
PGDB_AS002511
View
IC50
-
=
1
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A028389
PGDB_C008002
PGDB_AS002511
View
IC50
-
=
1
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A029177
PGDB_C008019
PGDB_AS002511
View
IC50
-
=
1
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A029721
PGDB_C008012
PGDB_AS002511
View
IC50
-
=
1
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A030041
PGDB_C008011
PGDB_AS002511
View
IC50
-
=
1
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A031187
PGDB_C008008
PGDB_AS002511
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A034425
PGDB_C008003
PGDB_AS002511
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A036098
PGDB_C008001
PGDB_AS002511
View
IC50
-
=
1
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A036770
PGDB_C008010
PGDB_AS002511
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A037774
PGDB_C007999
PGDB_AS002511
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A040522
PGDB_C007976
PGDB_AS002511
View