Summary
AssigneeBaifang Cayman
Filing years2023
Patents1
Compounds28
Activity records67
Patent families1
Targets1
Assay familiesdegradation, viability
Activity metricsIC50, degradation
Overview

Target distribution and active-compound trend

Target distribution

67 activity records

1 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

014282025
Activity compounds and values

Activity records

67 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C002859
% Degradation-=40%--GSPT1-HL-60WO2024073871A1PGDB_A009692PGDB_C002859PGDB_AS000569View
2D structure for PGDB_C002877
IC50-=9.2nM-GSPT1-HL-60WO2024073871A1PGDB_A010092PGDB_C002877PGDB_AS000219View
2D structure for PGDB_C002869
% Degradation-=0%--GSPT1-HL-60WO2024073871A1PGDB_A012950PGDB_C002869PGDB_AS000569View
2D structure for PGDB_C002852
% Degradation-=30%--GSPT1-HL-60WO2024073871A1PGDB_A017711PGDB_C002852PGDB_AS000569View
2D structure for PGDB_C002876
IC50-=23nM-GSPT1-HL-60WO2024073871A1PGDB_A017879PGDB_C002876PGDB_AS000219View
2D structure for PGDB_C002853
% Degradation-=0%--GSPT1-HL-60WO2024073871A1PGDB_A020268PGDB_C002853PGDB_AS001173View
2D structure for PGDB_C002877
% Degradation-=95%--GSPT1-HL-60WO2024073871A1PGDB_A022297PGDB_C002877PGDB_AS001173View
2D structure for PGDB_C002851
% Degradation-=0%--GSPT1-HL-60WO2024073871A1PGDB_A022945PGDB_C002851PGDB_AS001173View
2D structure for PGDB_C002857
% Degradation-=63%--GSPT1-HL-60WO2024073871A1PGDB_A023659PGDB_C002857PGDB_AS001173View
2D structure for PGDB_C002871
% Degradation-=29%--GSPT1-HL-60WO2024073871A1PGDB_A023672PGDB_C002871PGDB_AS001173View
2D structure for PGDB_C002865
% Degradation-=32%--GSPT1-HL-60WO2024073871A1PGDB_A023676PGDB_C002865PGDB_AS001173View
2D structure for PGDB_C002872
% Degradation-=33%--GSPT1-HL-60WO2024073871A1PGDB_A023723PGDB_C002872PGDB_AS000569View
2D structure for PGDB_C002870
% Degradation-=40%--GSPT1-HL-60WO2024073871A1PGDB_A023810PGDB_C002870PGDB_AS001173View
2D structure for PGDB_C002864
IC50-=290nM-GSPT1-HL-60WO2024073871A1PGDB_A023978PGDB_C002864PGDB_AS000219View
2D structure for PGDB_C002855
% Degradation-=52%--GSPT1-HL-60WO2024073871A1PGDB_A024451PGDB_C002855PGDB_AS001173View
2D structure for PGDB_C002876
% Degradation-=90%--GSPT1-HL-60WO2024073871A1PGDB_A027064PGDB_C002876PGDB_AS001173View
2D structure for PGDB_C002850
% Degradation-=45%--GSPT1-HL-60WO2024073871A1PGDB_A027843PGDB_C002850PGDB_AS000569View
2D structure for PGDB_C002855
% Degradation-=46%--GSPT1-HL-60WO2024073871A1PGDB_A029710PGDB_C002855PGDB_AS000569View
2D structure for PGDB_C002865
% Degradation-=26%--GSPT1-HL-60WO2024073871A1PGDB_A031282PGDB_C002865PGDB_AS000569View
2D structure for PGDB_C002858
% Degradation-=15%--GSPT1-HL-60WO2024073871A1PGDB_A031542PGDB_C002858PGDB_AS001173View