PatGlueDB | Molecular Glue Patent Bioactivity Database

Activity compounds and values

Activity records

36 records

	Control		Value		Concentration	Time					Record ID	Compound	Assay	Details
IC50	-	=	30.35	nM	-	—	CDK12	-	MDA-MB-231	CN121108130A	PGDB_A008061	PGDB_C007331	PGDB_AS001069	View
IC50	-	=	19.37	nM	-	—	CDK12	-	-	CN121108130A	PGDB_A008223	PGDB_C007326	PGDB_AS002060	View
IC50	-	=	57.46	nM	-	—	CDK12	-	-	CN121108130A	PGDB_A008550	PGDB_C007335	PGDB_AS002060	View
IC50	-	>	10000	nM	-	—	CDK12	-	MDA-MB-468	CN121108130A	PGDB_A009020	PGDB_C007327	PGDB_AS000556	View
IC50	-	=	31.52	nM	-	—	CDK12	-	-	CN121108130A	PGDB_A010946	PGDB_C007328	PGDB_AS002060	View
IC50	-	=	20.28	nM	-	—	CDK12	-	MDA-MB-468	CN121108130A	PGDB_A012172	PGDB_C007164	PGDB_AS000556	View
IC50	-	=	2861	nM	-	—	CDK12	-	MDA-MB-231	CN121108130A	PGDB_A013315	PGDB_C007327	PGDB_AS001069	View
IC50	-	=	10.11	nM	-	—	CDK12	-	MDA-MB-468	CN121108130A	PGDB_A019437	PGDB_C007325	PGDB_AS000556	View
IC50	-	=	13.5	nM	-	—	CDK12	-	MDA-MB-468	CN121108130A	PGDB_A020953	PGDB_C007331	PGDB_AS000556	View
IC50	-	>	10000	nM	-	—	CDK12	-	-	CN121108130A	PGDB_A022810	PGDB_C007333	PGDB_AS002060	View
IC50	-	=	34.54	nM	-	—	CDK12	-	-	CN121108130A	PGDB_A028513	PGDB_C007325	PGDB_AS002060	View
IC50	-	=	351.6	nM	-	—	CDK12	-	MDA-MB-231	CN121108130A	PGDB_A031323	PGDB_C007329	PGDB_AS001069	View
IC50	-	=	17.51	nM	-	—	CDK12	-	-	CN121108130A	PGDB_A031523	PGDB_C007331	PGDB_AS002060	View
IC50	-	=	219	nM	-	—	CDK12	-	MDA-MB-231	CN121108130A	PGDB_A033466	PGDB_C007335	PGDB_AS001069	View
IC50	-	=	2925	nM	-	—	CDK12	-	MDA-MB-231	CN121108130A	PGDB_A035112	PGDB_C007333	PGDB_AS001069	View
IC50	-	=	36.24	nM	-	—	CDK12	-	MDA-MB-468	CN121108130A	PGDB_A036721	PGDB_C007330	PGDB_AS000556	View
IC50	-	=	46.44	nM	-	—	CDK12	-	MDA-MB-231	CN121108130A	PGDB_A040486	PGDB_C007326	PGDB_AS001069	View
IC50	-	=	353.7	nM	-	—	CDK12	-	MDA-MB-468	CN121108130A	PGDB_A044111	PGDB_C007335	PGDB_AS000556	View
IC50	-	>	10000	nM	-	—	CDK12	-	MDA-MB-468	CN121108130A	PGDB_A048055	PGDB_C007333	PGDB_AS000556	View
IC50	-	=	196.5	nM	-	—	CDK12	-	MDA-MB-468	CN121108130A	PGDB_A050347	PGDB_C007332	PGDB_AS000556	View

Rows per pagePage 1 of 2 · 36 recordsGo to page

Zhongke Zhongshan Pharmaceutical Innovation Research Institute

Target distribution and active-compound trend

Target distribution

Active compounds by publication year

Activity records