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Compound
PGDB_C002812
8 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(NC(=O)c4cccc(C(=O)c5ccccc5)c4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 84 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A010621 | PGDB_C002812 | PGDB_AS000768 | View |
| % Degradation | - | = | 9 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A015285 | PGDB_C002812 | PGDB_AS002431 | View |
| % Degradation | - | = | 59.5 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A019474 | PGDB_C002812 | PGDB_AS000707 | View |
| % Degradation | - | = | 69.8 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A031991 | PGDB_C002812 | PGDB_AS000685 | View |
| % Degradation | - | = | 93.9 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A043910 | PGDB_C002812 | PGDB_AS000892 | View |
| % Degradation | - | = | 82.6 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A044609 | PGDB_C002812 | PGDB_AS001414 | View |
| % Degradation | - | = | 13.7 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A048582 | PGDB_C002812 | PGDB_AS001974 | View |
| % Degradation | - | = | 63.7 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A075398 | PGDB_C002812 | PGDB_AS000209 | View |