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Compound
PGDB_C002817
8 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(NC(=O)C4=COc5ccccc5O4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 70.8 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A008495 | PGDB_C002817 | PGDB_AS001414 | View |
| % Degradation | - | = | 90.7 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A014327 | PGDB_C002817 | PGDB_AS000892 | View |
| % Degradation | - | = | 35.2 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A015293 | PGDB_C002817 | PGDB_AS000768 | View |
| % Degradation | - | = | 1.2 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A015763 | PGDB_C002817 | PGDB_AS001974 | View |
| % Degradation | - | = | 60.3 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A034940 | PGDB_C002817 | PGDB_AS000685 | View |
| % Degradation | - | = | -0.1 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A035242 | PGDB_C002817 | PGDB_AS002431 | View |
| % Degradation | - | = | 13.4 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A050546 | PGDB_C002817 | PGDB_AS000707 | View |
| % Degradation | - | = | 46.4 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A059069 | PGDB_C002817 | PGDB_AS000209 | View |