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Compound
PGDB_C002819
8 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(NC(=O)c4ccc5occc5c4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 50.2 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A009085 | PGDB_C002819 | PGDB_AS000209 | View |
| % Degradation | - | = | 4.4 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A055712 | PGDB_C002819 | PGDB_AS001974 | View |
| % Degradation | - | = | 61.1 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A064349 | PGDB_C002819 | PGDB_AS001414 | View |
| % Degradation | - | = | 6.4 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A067873 | PGDB_C002819 | PGDB_AS000707 | View |
| % Degradation | - | = | 22.3 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A068128 | PGDB_C002819 | PGDB_AS000768 | View |
| % Degradation | - | = | 64.7 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A070081 | PGDB_C002819 | PGDB_AS000685 | View |
| % Degradation | - | = | 90.6 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A075522 | PGDB_C002819 | PGDB_AS000892 | View |
| % Degradation | - | = | 2 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A075620 | PGDB_C002819 | PGDB_AS002431 | View |