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Compound
PGDB_C002821
8 activity records1 related patents
2D structure
COc1ccc2c(CC(=O)Nc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)cccc2c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 57 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A010956 | PGDB_C002821 | PGDB_AS000685 | View |
| % Degradation | - | = | 97.7 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A016752 | PGDB_C002821 | PGDB_AS000707 | View |
| % Degradation | - | = | 98.4 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A016965 | PGDB_C002821 | PGDB_AS000768 | View |
| % Degradation | - | = | 29 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A019114 | PGDB_C002821 | PGDB_AS002431 | View |
| % Degradation | - | = | 93 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A029613 | PGDB_C002821 | PGDB_AS001414 | View |
| % Degradation | - | = | 63.4 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A041166 | PGDB_C002821 | PGDB_AS000209 | View |
| % Degradation | - | = | 41.9 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A050704 | PGDB_C002821 | PGDB_AS001974 | View |
| % Degradation | - | = | 95.8 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A053612 | PGDB_C002821 | PGDB_AS000892 | View |