Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C002822
8 activity records1 related patents
2D structure
COc1ccc2cccc(CC(=O)Nc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)c2c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 21.3 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A018887 | PGDB_C002822 | PGDB_AS001974 | View |
| % Degradation | - | = | 64.4 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A035685 | PGDB_C002822 | PGDB_AS000685 | View |
| % Degradation | - | = | 97.6 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A037673 | PGDB_C002822 | PGDB_AS000768 | View |
| % Degradation | - | = | 96.9 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A062097 | PGDB_C002822 | PGDB_AS000707 | View |
| % Degradation | - | = | 92.2 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A065548 | PGDB_C002822 | PGDB_AS001414 | View |
| % Degradation | - | = | 16.6 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A071078 | PGDB_C002822 | PGDB_AS002431 | View |
| % Degradation | - | = | 94.4 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A072024 | PGDB_C002822 | PGDB_AS000892 | View |
| % Degradation | - | = | 59.7 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A076179 | PGDB_C002822 | PGDB_AS000209 | View |